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25 Years of Small-Molecule Optimization at Novartis: A Retrospective Analysis of Chemical Series Evolution.
Maximilian Beckers
Nikolas Fechner
Nikolaus Stiefl
Published in:
J. Chem. Inf. Model. (2022)
Keyphrases
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drug discovery
global optimization
optimization problems
years ago
optimization process
constrained optimization
search engine
optimal design
temporal evolution
real world
image sequences
lower bound
optimization algorithm
optimization methods
small size
chemical compounds